Process for preparing spray dried formulations of 4-[[6-amino-5-bromo-2-[(4-cyanophenyl)amino]-4-pyrimidinyl]oxy]-3,5-dimethylbenzonitrile
US9603803B2 · kind B2 · utility
0Cited by
2References
9Claims
0Family size
Assignee
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Key dates
| Filing date | Feb 16, 2012 |
| Grant date | Mar 28, 2017 |
| Priority date | — |
| Expiry date | Feb 16, 2032 |
Classification
- Technology area (CPC A)Human Necessities
- CPC primaryA61P31/18
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
This invention relates to a process for producing a spray-dried powder comprising microcrystalline cellulose in a solid dispersion of the anti-HIV compound etravirine (TMC125) in a water-soluble polymer.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.