Patent · US Active

Azetidinyl phenyl, pyridyl or pyrazinyl carboxamide derivatives as JAK inhibitors

US9611269B2 · kind B2 · utility

41Cited by
80References
24Claims
0Family size

Assignee

Inventors

Key dates

Filing dateApr 27, 2015
Grant dateApr 4, 2017
Priority date
Expiry dateApr 27, 2035

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D471/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides azetidinyl phenyl, pyridyl, or pyrazinyl carboxamide derivatives, as well as their compositions and methods of use, that modulate the activity of Janus kinase (JAKs) and are useful in the treatment of diseases related to the activity of JAK including, for example, inflammatory disorders, autoimmune disorders, cancer, and other diseases.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.