Patent · US Active

Pharmaceutical formulations of a Bruton's tyrosine kinase inhibitor

US9655857B2 · kind B2 · utility

22Cited by
79References
37Claims
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Key dates

Filing dateMar 3, 2016
Grant dateMay 23, 2017
Priority date
Expiry dateMar 3, 2036

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Described herein are pharmaceutical formulations of Bruton's tyrosine kinase (Btk) inhibitor 1-((R)-3-(4-amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one. Also disclosed are methods of using the Btk inhibitor, alone or in combination with other therapeutic agents, for the treatment of autoimmune diseases or conditions, heteroimmune diseases or conditions, cancer, including lymphoma, and inflammatory diseases or conditions.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.