Patent · US Active

Aminopyrimidinyl compounds

US9663526B2 · kind B2 · utility

9Cited by
3References
26Claims
0Family size

Assignee

Inventors

Key dates

Filing dateAug 19, 2015
Grant dateMay 30, 2017
Priority date
Expiry dateAug 19, 2035

Classification

  • Technology area (CPC H)Electricity
  • CPC primaryH04N7/188
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A compound having the structure:or an acceptable salt thereof, wherein X is N or CR, where R is hydrogen, alkyl, etc.; A is selected from the group consisting of a bond, C═O, —SO2—, etc.; A′ is selected from the group consisting of a bond, C═O, etc.; Z is —(CH2)h— or a bond, etc.; R1 and R1′ are independently selected from the group consisting of hydrogen, alkyl, etc.; R2 is selected from hydrogen, alkyl, etc.; R3 is selected from the group consisting of hydrogen, and amino; R4 is monocyclic or bicyclic, etc.; R5 is independently selected from hydrogen, alkyl, etc.; h, j, k, m, n and q are integers as defined in the specification. Also provided are methods of treatment as Janus Kinase inhibitors and pharmaceutical compositions containing the compounds of the invention and combinations with other therapeutic agents.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.