Patent · US Active

Alpha-amino boronic acid derivatives, selective immunoproteasome inhibitors

US9688702B2 · kind B2 · utility

2Cited by
1References
16Claims
0Family size

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Inventors

Key dates

Filing dateDec 21, 2012
Grant dateJun 27, 2017
Priority date
Expiry dateMay 10, 2033

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07F5/02
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides compounds of Formula (I) as inhibitors of LMP7 for the treatment of autoimmune and inflammatory diseases.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.