Patent · US Active

Cephem compounds, their production and use

US9751894B2 · kind B2 · utility

1Cited by
9References
12Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 5, 2016
Grant dateSep 5, 2017
Priority date
Expiry dateDec 5, 2036

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D501/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Cephem compounds, pharmaceutically acceptable salts thereof, and methods of using same, wherein the compound has a bicyclic nitrogen-containing aromatic heterocyclic ring as the quaternary ammoniomethyl group at the 3-position and one or both of a terminal amidine residue (substituted or unsubstituted) attached to an aryl or a 5- or 6-membered heteroaryl group (substituted or unsubstituted) which is further attached through a spacer to the free N-atom of the quaternary nitrogen-containing bicyclic ring at the 3-side chain, or a terminal guanidine residue attached to an aryl or a 5- or 6-membered heteroaryl group (substituted or unsubstituted) which is further attached through a spacer to the free N-atom of the quaternary nitrogen-containing bicyclic ring at the 3-side chain.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.