Patent · US Active

Labeled iodinated tropane formulation

US9757483B2 · kind B2 · utility

0Cited by
19References
1Claims
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Key dates

Filing dateOct 17, 2014
Grant dateSep 12, 2017
Priority date
Expiry dateOct 17, 2034

Classification

  • Technology area (CPC G)Physics
  • CPC primaryG21H5/02
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A diagnostic formulation is provided comprising a tropane having a radioactive concentration of at least 1.6 mCi/mL at least about 51 hours post creation. The diagnostic formulation optionally comprises a radiolabeled dopamine transporter (DAT) ligand useful in the diagnosis of Parkinson's disease (PS). One example of a radiolabeled dopamine transporter (DAT) ligand example is [123I]-2β-carbomethoxy-3β-(4-flurophenyl)-N-(3-iodo-E-allyl) nortropane.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.