Patent · US Active

Alvocidib prodrugs having increased bioavailability

US9758539B2 · kind B2 · utility

22Cited by
7References
13Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 18, 2016
Grant dateSep 12, 2017
Priority date
Expiry dateMay 18, 2036

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D405/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds having the following structure (I):or a stereoisomer, tautomer or pharmaceutically acceptable salt thereof, wherein one of R1, R2 or R3 is —P(═O)(OH)2, and the other two of R1, R2 and R3 are each H, are provided. Pharmaceutical compositions comprising the compounds, and methods for use of the compounds for treating diseases associated with overexpression of a cyclin-dependent kinase (CDK) are also provided.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.