Patent · US Active

Quinoxaline derivatives as GPR6 modulators

US9770452B2 · kind B2 · utility

2Cited by
0References
22Claims
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Assignee

Inventors

Key dates

Filing dateOct 25, 2016
Grant dateSep 26, 2017
Priority date
Expiry dateOct 25, 2036

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D471/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides compounds of Formula (I):that are GPR6 modulators and are therefore useful for the treatment of diseases treatable by modulation of GPR6, in particular treating Parkinson disease, levodopa induced dyskinesias, Huntington's disease, other dyskinesias, akinesias, and motor disorders involving dysfunction of the striatum, schizophrenia and drug addiction. Also provided are pharmaceutical compositions containing such compounds and processes for preparing such compounds.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.