Patent · US Active

Tricyclic inhibitors of HIF-2-alpha and uses thereof

US9796697B2 · kind B2 · utility

14Cited by
4References
18Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 8, 2016
Grant dateOct 24, 2017
Priority date
Expiry dateJun 8, 2036

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D409/12
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Compounds comprising a fused tricylic core that modulate HIF-2α activity, pharmaceutical compositions containing these chemical entities, and methods of using these chemical entities for treating diseases associated with HIF-2α activity are described herein.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.