α-glucosidase inhibitors

US9802894B2 · kind B2 · utility

Assignee

• KING SAUD UNIVERSITY · SA

Inventors

• Abdullah Mohammed Al-Majid · Riyadh, SA
• Mohammad Shahidul Islam · Riyadh, SA
• Assem Barakat · Riyadh, SA
• Muhammad Iqbal Choudhary · Karachi, PK
• Sammer Yousuf · Karachi, PK

Key dates

• Filing date: Sep 29, 2015
• Grant date: Oct 31, 2017
• Expiry date: Sep 29, 2035

Classification

• Technology area (CPC C): Chemistry; Metallurgy
• CPC primary: C07D209/12
• WIPO field: Organic fine chemistry
• WIPO sector: Chemistry

Abstract

Novel α-Glucosidase inhibitors include propanone substituted indole ring-containing heterocyclic compounds, which are represented by Formula I:WhereinR1 is thiophene, 2,4-di chloro phenyl, 2,6-di chloro phenyl, bromo phenyl, benzyl or nitrophenyl; and R2 is an aryl group, or stereoisomers or pharmaceutically acceptable salts thereof.