Patent · US Active

Process for the preparation of substituted cycloserines

US9815803B2 · kind B2 · utility

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4Claims
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Assignee

Inventors

Key dates

Filing dateApr 3, 2017
Grant dateNov 14, 2017
Priority date
Expiry dateApr 3, 2037

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D261/12
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention relates to processes for the preparation of substituted cycloserine compounds of formula (I)wherein R1 is C1-C8alkyl, C1-C8haloalkyl, C3-C6 cycloalkyl, aryl or aryl substituted by one to five R11, or aryl-C1-C4alkylene or aryl-C1-C4alkylene substituted by one to five R11; andeach R11 is independently C1-C4alkyl, C1-C4haloalkyl, C1-C4alkoxy, C1-C4haloalkoxy, cyano or halogen;The invention also relates to intermediates produced by the processes.Compounds of formula (I) are useful intermediates for the production of compounds in the agricultural and pharmaceutical fields.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.