Patent · US Active

Quinazolinones and azaquinazolinones as ubiquitin-specific protease 7 inhibitors

US9840491B2 · kind B2 · utility

21Cited by
60References
17Claims
0Family size

Assignee

Inventors

Key dates

Filing dateFeb 4, 2016
Grant dateDec 12, 2017
Priority date
Expiry dateFeb 4, 2036

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present disclosure relates to inhibitors of USP7 inhibitors useful in the treatment of cancers, neurodegenerative diseases, immunological disorders, inflammatory disorders, cardiovascular diseases, ischemic diseases, viral infections and diseases, and bacterial infections and diseases, having the Formula:where R1, R2, R3, R4, R4′, X1, Y1, Y2, Y3, Y4, n, and m are described herein.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.