Patent · US Active

Analogues of 4H-pyrazolo[1,5-a] benzimidazole compound as PARP inhibitors

US9856262B2 · kind B2 · utility

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21Claims
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Key dates

Filing dateMar 30, 2015
Grant dateJan 2, 2018
Priority date
Expiry dateMar 30, 2035

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D519/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Disclosed is a series of analogs of 4H-pyrazolo[1,5-α]benzimidazole compound as PARP inhibitors. In particular, disclosed in the invention is a compound as shown by formula (I) or a pharmaceutically acceptable salt thereof as a PARP inhibitor.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.