Analogues of 4H-pyrazolo[1,5-a] benzimidazole compound as PARP inhibitors
US9856262B2 · kind B2 · utility
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21Claims
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Key dates
| Filing date | Mar 30, 2015 |
| Grant date | Jan 2, 2018 |
| Priority date | — |
| Expiry date | Mar 30, 2035 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D519/00
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
Disclosed is a series of analogs of 4H-pyrazolo[1,5-α]benzimidazole compound as PARP inhibitors. In particular, disclosed in the invention is a compound as shown by formula (I) or a pharmaceutically acceptable salt thereof as a PARP inhibitor.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.