Patent · US Active

Stable pharmaceutical composition containing 8-[(3R)-3-amino-1-piperidinyl]-7-(2-butyn-1-yl)-3,7-dihydro-3-methyl-1-[(4-methyl-2-quinazolinyl)methyl]-1H-purine-2,6-dione or a pharmaceutically acceptable salt thereof

US9867829B2 · kind B2 · utility

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21Claims
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Assignee

Inventors

Key dates

Filing dateAug 12, 2013
Grant dateJan 16, 2018
Priority date
Expiry dateAug 12, 2033

Classification

  • Technology area (CPC B)Performing Operations; Transporting
  • CPC primaryB65D2565/388
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to a stable pharmaceutical composition comprising amorphous or crystalline linagliptin or a pharmaceutically acceptable salt of linagliptin, mannitol, copovidone, and magnesium stearate, processes for preparing the stable pharmaceutical composition, and a container comprising the stable pharmaceutical composition.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.