Stable pharmaceutical composition containing 8-[(3R)-3-amino-1-piperidinyl]-7-(2-butyn-1-yl)-3,7-dihydro-3-methyl-1-[(4-methyl-2-quinazolinyl)methyl]-1H-purine-2,6-dione or a pharmaceutically acceptable salt thereof
US9867829B2 · kind B2 · utility
0Cited by
0References
21Claims
0Family size
Assignee
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Key dates
| Filing date | Aug 12, 2013 |
| Grant date | Jan 16, 2018 |
| Priority date | — |
| Expiry date | Aug 12, 2033 |
Classification
- Technology area (CPC B)Performing Operations; Transporting
- CPC primaryB65D2565/388
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
The present invention relates to a stable pharmaceutical composition comprising amorphous or crystalline linagliptin or a pharmaceutically acceptable salt of linagliptin, mannitol, copovidone, and magnesium stearate, processes for preparing the stable pharmaceutical composition, and a container comprising the stable pharmaceutical composition.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.