Cyclic vinylogous amides as bromodomain inhibitors
US9884806B2 · kind B2 · utility
0Cited by
4References
20Claims
0Family size
Assignee
Inventors
Key dates
| Filing date | Aug 29, 2014 |
| Grant date | Feb 6, 2018 |
| Priority date | — |
| Expiry date | Aug 29, 2034 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D295/21
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
Cyclic vinylogous amides of Formula I are disclosedThe compounds are useful for treating diseases that arise from inappropriate activity of proteins containing an acetyl-lysine. The compositions comprise a genus of cyclic vinylogous amides that are inhibitors of bromodomain.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.