Patent · US Active

Polymorphs of ARRY-380, a selective HER 2 inhibitor and pharmaceutical compositions containing them

US9889134B2 · kind B2 · utility

7Cited by
3References
16Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 26, 2015
Grant dateFeb 13, 2018
Priority date
Expiry dateOct 26, 2035

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D471/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Polymorphs of N4-(4-([1,2,4]triazolo[1,5-a]pyridin-7-yloxy)-3-methylphenyl)-N6-(4,4-dimethyl-4,5-dihydrooxazol-2-yl)quinazoline-4,6-diamine are provided herein. Processes for preparing the polymorphs and pharmaceutical composition comprising the polymorphs are also disclosed.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.