Patent · US Active

Polysubstituted pyridine compound, preparation method, use and pharmaceutical composition

US9902709B2 · kind B2 · utility

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4Claims
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Key dates

Filing dateDec 30, 2014
Grant dateFeb 27, 2018
Priority date
Expiry dateDec 30, 2034

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P35/02
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides a polysubstituted pyridine compound of Formula I, a preparation method, a use and a pharmaceutical composition thereof. The polysubstituted pyridine compound of Formula I according to the present invention has an excellent anti-tumor effect, can inhibit various cell kinases simultaneously, has significantly excellent pharmacokinetic characteristics, and is very suitable for oral and intravenous administration. The pharmaceutical composition according to the present invention can be useful for treating tumors and cancers.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.