Patent · US Active

Heterocyclic derivatives as RORgamma modulators

US9902725B2 · kind B2 · utility

3Cited by
2References
19Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 22, 2015
Grant dateFeb 27, 2018
Priority date
Expiry dateDec 22, 2035

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D403/12
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention provides novel compounds of formula (I) that are modulators of RORgamma. These compounds, and pharmaceutical compositions comprising the same, are suitable means for treating any disease wherein the modulation of RORgamma has therapeutic effects, for instance in autoimmune diseases, autoimmune-related diseases, inflammatory diseases, fibrotic diseases, or cholestatic diseases.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.