Patent · US Active

Methods of synthesizing a difluorolactam analog

US9914725B2 · kind B2 · utility

0Cited by
7References
4Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 14, 2014
Grant dateMar 13, 2018
Priority date
Expiry dateMar 14, 2034

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07F9/4006
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention relates to processes and intermediates for preparing compounds of formula (IA), wherein R1, R4, R5, R6, and L1 are as defined herein. Compounds of formula (IA) have been found useful as EP4 receptor agonists useful in the treatment of glaucoma, osteoporosis, neuropathic pain, and related disorders.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.