Patent · US Active

Method of treating estrogen receptor (ER)-positive breast cancers with selective androgen receptor modulator (SARMS)

US9969683B2 · kind B2 · utility

2Cited by
77References
9Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 29, 2013
Grant dateMay 15, 2018
Priority date
Expiry dateJan 22, 2035

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C237/20
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

This invention relates to the treatment of breast cancer in a subject, for example a female subject. The breast cancer includes metastatic breast cancer, refractory breast cancer, AR-positive breast cancer, AR-positive refractory breast cancer, AR-positive metastatic breast cancer, AR-positive and ER-positive breast cancer, triple negative breast cancer, advanced breast cancer, breast cancer that has failed SERM (tamoxifen, toremifene), aromatase inhibitor, trastuzumab (Herceptin, ado-trastuzumab emtansine), pertuzumab (Perjeta), lapatinib, exemestane (Aromasin), bevacizumab (Avastin), and/or fulvestrant treatments, and metastasis in a subject suffering from breast cancer. The method comprises administering to the subject a therapeutically effective amount of a selective androgen receptor modulator (SARM) compound.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.