Patent · US Active

Fused bicyclic heteroaromatic derivatives as kinase inhibitors

US9969748B2 · kind B2 · utility

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Key dates

Filing dateJun 11, 2015
Grant dateMay 15, 2018
Priority date
Expiry dateJun 11, 2035

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02A50/30
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A series of fused bicyclic heteroaromatic derivatives of formula (IA) or (IB), as defined herein, being selective inhibitors of phosphatidylinositol-4-kinase IIIβ (PI4KIIIβ) activity, are beneficial in the treatment and/or prevention of various human ailments, including inflammatory, autoimmune and oncological disorders; viral diseases and malaria; and organ and cell transplant rejection.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.