Patent · US Active

Cannabinoid receptor antagonists/inverse agonists useful for treating metabolic disorders, including obesity and diabetes

US9987253B2 · kind B2 · utility

7Cited by
9References
19Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 13, 2016
Grant dateJun 5, 2018
Priority date
Expiry dateDec 13, 2036

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D231/06
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides novel, diastereomeric pyrazolines that are useful as cannabinoid receptor blockers and pharmaceutical compositions thereof and methods of using the same for treating obesity, diabetes, inflammatory disorders, cardiometabolic disorders, hepatic disorders, and/or cancers.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.