Inventor · Baltimore, MD, US

Alexander D. MACKERELL, JR.

28Patents
5h-index
38Co-inventors
69Inventor score

Filing activity: Jul 31, 2001 → Oct 18, 2024

Most-cited inventions

PatentTitleAreaCited byStatus
US8338464B2 Small molecule inhibitors of BCL6 Chemistry; Metallurgy 27 Active
US11078171B2 Non-ATP/catalytic site p38 mitogen activated protein kinase inhibitors Chemistry; Metallurgy 11 Active
US11357781B2 Non-catalytic substrate-selective, p38α-specific MAPK inhibitors with endothelial-stabilizing and anti-inflammatory activity, and methods of use thereof Chemistry; Metallurgy 7 Active
US7915245B2 Methods and compositions of trail-death receptor agonists/activators Human Necessities 7 Active
US9115122B2 Non-ATP dependent inhibitors of extracellular signal-regulated kinase (ERK) Chemistry; Metallurgy 5 Active
US8785499B2 Targeting NAD biosynthesis in bacterial pathogens Human Necessities 3 Active
US8796323B2 Defensin-like molecules as novel antimicrobial agents Human Necessities 3 Active
US8445537B2 Compounds that inhibit human DNA ligases and methods of treating cancer Physics 3 Active
US11718595B2 Non-ATP/catalytic site p38 Mitogen Activated Protein Kinase inhibitors Chemistry; Metallurgy 2 Active
US9351963B2 Defensin-like molecules as novel antimicrobial agents Human Necessities 2 Active
US9073896B2 Compounds that inhibit human DNA ligases and methods of treating cancer Physics 1 Active
US7521463B2 Immunomodulatory compounds Human Necessities 1 Expired
US11911392B2 Non-catalytic substrate-selective p38α-specific MAPK inhibitors with endothelial-stabilizing and anti-inflammatory activity, and methods of use thereof Chemistry; Metallurgy 0 Active
US12404259B2 Inhibitors of extracellular signal-regulated kinase Human Necessities 0 Active
US9757375B2 Compounds that inhibit human DNA ligases and methods of treating cancer Physics 0 Active
US8053477B2 Inhibitors of the S100-p53 protein-protein interaction and method of inhibiting cancer employing the same Human Necessities 0 Expired
US10941114B2 Small molecule lipid II inhibitors Chemistry; Metallurgy 0 Active
US10961214B2 Small molecule lipid II inhibitors Chemistry; Metallurgy 0 Active
US11911393B2 Non-catalytic substrate-selective p38alpha-specific MAPK inhibitors with endothelial-stabilizing and anti-inflammatory activity, and methods of use thereof Chemistry; Metallurgy 0 Active
US8476273B2 Small molecule inhibitors of Lck SH2 domain binding Human Necessities 0 Active
US12202810B2 Non-ATP/catalytic site p38 mitogen activated protein kinase inhibitors Chemistry; Metallurgy 0 Active
US9701627B2 LRRK2 GTP binding inhibitors for treatment of Parkinson's disease and neuroinflammatory disorders Chemistry; Metallurgy 0 Active
US9422302B2 Mixed μ agonist/ δ antagonist opioid analgesics with reduced tolerance liabilities and uses thereof Chemistry; Metallurgy 0 Active
US11510908B2 Protein translation inhibitors and uses thereof Human Necessities 0 Active
US11634381B2 RUNX2 transcription factor inhibitors and uses thereof Chemistry; Metallurgy 0 Active

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.