Inventor · North Wales, PA, US

Mark E. Fraley

68Patents
16h-index
99Co-inventors
87Inventor score

Filing activity: Jun 24, 1996 → Dec 4, 2017

Most-cited inventions

PatentTitleAreaCited byStatus
US7550470B2 Substituted pyrazolo[1,5-A]pyrimidines as tyrosine kinase inhibitors Human Necessities 92 Expired
US6306874A Tyrosine kinase inhibitors Chemistry; Metallurgy 70 Expired
US6235741A Angiogenesis inhibitors Chemistry; Metallurgy 46 Expired
US6245759A Tyrosine kinase inhibitors Human Necessities 44 Expired
US5668289A Pyridinone thrombin inhibitors Human Necessities 34 Expired
US6265403A Angiogenesis inhibitors Human Necessities 31 Expired
US6313138A Tyrosine kinase inhibitors Human Necessities 31 Expired
US6479512B1 Tyrosine kinase inhibitors Chemistry; Metallurgy 29 Expired
US6420382B2 Tyrosine kinase inhibitors Human Necessities 29 Expired
US5872138A Thrombin inhibitors Chemistry; Metallurgy 24 Expired
US8623863B2 Disubstituted azepan orexin receptor antagonists Chemistry; Metallurgy 23 Active
US7262187B2 Substituted oxazolo- and thizaolopyrimidinones as a mitotic kinesin inhibitor Human Necessities 20 Expired
US7192949B2 Substituted bicyclic pyrimidinones as a mitotic kinesin KSP inhibitors Chemistry; Metallurgy 19 Expired
US8754096B2 Piperidinone carboxamide azaindane CGRP receptor antagonists Chemistry; Metallurgy 17 Active
US8912210B2 Piperidinone carboxamide azaindane CGRP receptor antagonists Chemistry; Metallurgy 17 Active
US8481556B2 Piperidinone carboxamide azaindane CGRP receptor antagonists Chemistry; Metallurgy 17 Active
US8883807B2 Piperidinone carboxamide indane CGRP receptor antagonists Chemistry; Metallurgy 15 Active
US6380203B1 Angiogenesis inhibitors Chemistry; Metallurgy 14 Expired
US9499545B2 Piperidinone carboxamide azaindane CGRP receptor antagonists Chemistry; Metallurgy 14 Active
US9833448B2 Piperidinone carboxamide azaindane CGRP receptor antagonists Chemistry; Metallurgy 13 Active
US9227972B2 Aliphatic spirolactam CGRP receptor antagonists Human Necessities 13 Active
US9227973B2 Pyridine CGRP receptor antagonists Chemistry; Metallurgy 12 Active
US9499541B2 Piperidinone carboxamide indane CGRP receptor antagonists Chemistry; Metallurgy 12 Active
US9296750B2 Spirolactam CGRP receptor antagonists Chemistry; Metallurgy 12 Active
US6544988B1 Tyrosine kinase inhibitors Human Necessities 12 Expired

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.