Inventor · Libertyville, IL, US

Megumi Kawai

25Patents
11h-index
35Co-inventors
75Inventor score

Filing activity: Dec 27, 1990 → Oct 18, 2010

Most-cited inventions

PatentTitleAreaCited byStatus
US5457111A Macrocyclic immunomodulators Chemistry; Metallurgy 95 Expired
US7772231B2 Substituted pyrazolo[3,4-d]pyrimidines as protein kinase inhibitors Human Necessities 62 Active
US6323228A 3-substituted indole angiogenesis inhibitors Chemistry; Metallurgy 58 Expired
US6242494A Substituted .beta.-amino acid inhibitors of methionine aminopeptidase-2 Chemistry; Metallurgy 29 Expired
US7030262B2 3-Amino-2-hydroxyalkanoic acids and their prodrugs Chemistry; Metallurgy 28 Expired
US5604294A Macrocyclic immunomodulators Chemistry; Metallurgy 25 Expired
US7491718B2 Sulfonamides having antiangiogenic and anticancer activity Chemistry; Metallurgy 25 Expired
US5457194A Substituted aliphatic amine-containing macrocyclic immunomodulators Human Necessities 19 Expired
US6887863B2 Hydrazide and alkoxyamide angiogenesis inhibitors Chemistry; Metallurgy 16 Expired
US5223485A Anaphylatoxin-receptor ligands Human Necessities 13 Expired
US5541189A Substituted aliphatic amine-containing macrocyclic immunomodulators Chemistry; Metallurgy 13 Expired
US6121257A Sulfamate containing macrocyclic immunomodulators Human Necessities 11 Expired
US5561228A Macrocyclic immunomodulators Chemistry; Metallurgy 11 Expired
US5708002A Macrocyclic immunomodulators Chemistry; Metallurgy 10 Expired
US5541193A Heterocycle-containing macrocyclic immunomodulators Chemistry; Metallurgy 9 Expired
US5561140A Substituted alicyclic amine-containing macrocyclic immunomodulators Human Necessities 9 Expired
US5530120A Substituted alicyclic aliphatic-amine containing macrocyclic immunomodulators Chemistry; Metallurgy 8 Expired
US5386011A Hexapeptide anaphylatoxin-receptor ligands Human Necessities 7 Expired
US5190922A Terminally modified tri-, tetra- and pentapeptide anaphylatoxin receptor ligands Human Necessities 7 Expired
US5530119A Substituted alicyclic amine-containing macrocyclic immunomodulators Human Necessities 6 Expired
US5387671A Hexa- and heptapeptide anaphylatoxin-receptor ligands Human Necessities 5 Expired
US6632961B1 Antiangiogenic drug to treat cancer, arthritis and retinopathy Chemistry; Metallurgy 5 Expired
US5561139A Substituted alicyclic-aliphatic amine-containing macrocyclic immunomodulators Chemistry; Metallurgy 5 Expired
US6849757B2 Antiangiogenic drug to treat cancer, arthritis and retinopathy Chemistry; Metallurgy 4 Expired
US9051315B2 Imidazopyridines as a novel scaffold for multi-targeted kinase inhibition Human Necessities 0 Active

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.