Inventor · Cambridge, GB

Miles Stuart Congreve

93Patents
14h-index
122Co-inventors
87Inventor score

Filing activity: Dec 16, 1999 → Mar 24, 2023

Most-cited inventions

PatentTitleAreaCited byStatus
US9670183B2 Bicyclic AZA compounds as muscarinic M1 receptor and/or M4 receptor agonists Chemistry; Metallurgy 30 Active
US6867192B1 Compounds useful in the treatment of inflammatory diseases Human Necessities 27 Expired
US8685980B2 Pyrrolopyrimidine compounds and their uses Human Necessities 27 Active
US8895745B2 Bicyclic heterocyclic compounds as FGFR inhibitors Chemistry; Metallurgy 24 Active
US9758506B2 Muscarinic agonists Human Necessities 21 Active
US9266857B2 Bicyclic AZA compounds as muscarinic M1 receptor agonists Chemistry; Metallurgy 20 Active
US9593106B2 Piperidin-1-yl and azepin-1-yl carboxylates as muscarinic M4 receptor agonists Chemistry; Metallurgy 20 Active
US10196380B2 Bicyclic aza compounds as muscarinic M1 receptor and/or M4 receptor agonists Chemistry; Metallurgy 16 Active
US7700625B2 Hydroxybenzamide derivatives and their use as inhibitors of Hsp90 Chemistry; Metallurgy 15 Active
US10112923B2 1,2,4-triazine-4-amine derivatives Chemistry; Metallurgy 15 Active
US9926297B2 Bicyclic AZA compounds as muscarinic M1 receptor and/or M4 receptor agonists Chemistry; Metallurgy 15 Active
US9187451B2 Muscarinic M1 receptor agonists Chemistry; Metallurgy 14 Active
US9669013B2 Bicyclic aza compounds as muscarinic M1 receptor agonists Chemistry; Metallurgy 14 Active
US8131527B1 FGFR pharmacophore compounds Physics 14 Active
US10259787B2 Substituted cyclohexanes as muscarinic M1 receptor and/or M4 receptor agonists Chemistry; Metallurgy 13 Active
US9907805B2 Muscarinic M1 receptor agonists Chemistry; Metallurgy 13 Active
US10385039B2 Bicyclic aza compounds as muscarnic M1 receptor and/or M4 receptor antagonists Chemistry; Metallurgy 12 Active
US8101648B2 Hydroxybenzamide derivatives and their use as inhibitors of HSP90 Chemistry; Metallurgy 12 Active
US7754725B2 Dihydroxyphenyl isoindolymethanones Chemistry; Metallurgy 12 Active
US10329278B2 Pharmaceutical compounds Chemistry; Metallurgy 12 Active
US8106057B2 Dihydroxyphenyl isoindolylmethanones Chemistry; Metallurgy 12 Active
US10759751B2 Substituted spirocyclohexanes as muscarinic M1 receptor and/or M4 receptor agonists Chemistry; Metallurgy 12 Active
US10689368B2 Bicyclic aza compounds as muscarinic M1 receptor and/or M4 receptor Chemistry; Metallurgy 11 Active
US9573929B2 Muscarinic M1 receptor agonists Chemistry; Metallurgy 11 Active
US10030035B2 Muscarinic receptor agonists Chemistry; Metallurgy 11 Active

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.