Inventor · Basel, CH

Vito Guagnano

33Patents
7h-index
60Co-inventors
68Inventor score

Filing activity: May 29, 2002 → Mar 15, 2021

Most-cited inventions

PatentTitleAreaCited byStatus
US8552002B2 Compounds and compositions as protein kinase inhibitors Chemistry; Metallurgy 77 Active
US8815901B2 Quinoline carboxamide derivatives as protein tyrosine kinase inhibitors Chemistry; Metallurgy 39 Active
US7652022B2 Diaryl urea derivatives useful for the treatment of protein kinase dependent diseases Chemistry; Metallurgy 13 Expired
US8293746B2 Pyrimidinyl aryl urea derivatives being FGF inhibitors Chemistry; Metallurgy 12 Active
US8759517B2 Pyrirnidinyl aryl urea derivatives being FGF inhibitors Chemistry; Metallurgy 9 Active
US8227462B2 Pyrrolidine-1,2-dicarboxamide derivatives Chemistry; Metallurgy 9 Active
US8969341B2 Pyrazolopyrrolidine compounds Human Necessities 7 Active
US8975417B2 Pyrazolopyrrolidine derivatives and their use in the treatment of disease Chemistry; Metallurgy 6 Active
US8815926B2 Substituted pyrrolo[3,4-D]imidazoles for the treatment of MDM2/4 mediated diseases Human Necessities 3 Active
US7795288B2 Thiazole and pyrazole derivatives as Flt-3 kinase inhibitors Chemistry; Metallurgy 3 Active
US8476268B2 Pyrrolidine-1,2-dicarboxamide derivatives Chemistry; Metallurgy 3 Active
US8030311B2 Phenylacetamides suitable as protein kinase inhibitors Chemistry; Metallurgy 1 Active
US7514447B2 Diarylamine-containing compounds and compositions, and their use as modulators of c-kit receptors Chemistry; Metallurgy 1 Active
US8710085B2 Pyrrolidine-1,2-dicarboxamide derivatives Chemistry; Metallurgy 1 Active
US9556180B2 Pyrazolo[3,4-d]pyrimidinone compounds as inhibitors of the P53/MDM2 interaction Human Necessities 1 Active
US9403827B2 Substituted purinone compounds Human Necessities 1 Active
US10028955B2 FGFR inhibitor for use in the treatment of hypophosphatemic disorders Human Necessities 1 Active
US9365576B2 Pyrrolopyrrolidinone compounds Human Necessities 1 Active
US7563894B2 Diarylamine-containing compounds and compositions, and their use as modulators of c-kit receptors Chemistry; Metallurgy 1 Active
US7592349B2 Diarylamine-containing compounds and compositions, and their use as modulators of c-kit receptors Chemistry; Metallurgy 1 Active
US7638523B2 Diarylamine-containing compounds and compositions, and their use as modulators of c-kit receptors Chemistry; Metallurgy 0 Active
US8273882B2 Quinoxaline carboxamide derivatives as protein tyrosine kinase inhibitors Chemistry; Metallurgy 0 Active
US6933290B2 2-{N-(2-amino-3-(heteroaryl or aryl)propionyl)-aminoacyl}-amino}-alkylboronic acid derivatives Human Necessities 0 Expired
US8859586B2 Cyclohexyl isoquinolinone compounds Chemistry; Metallurgy 0 Active
US12083101B2 Biaryl derivatives as YAP/TAZ-TEAD protein-protein interaction inhibitors Chemistry; Metallurgy 0 Active

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.