Patent · US Active

Heteroaryl pyridone and aza-pyrodine compounds

US10045983B2 · kind B2 · utility

6Cited by
11References
14Claims
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Key dates

Filing dateAug 31, 2017
Grant dateAug 14, 2018
Priority date
Expiry dateAug 31, 2037

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07F7/1804
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Heteroaryl pyridone and aza-pyridone compounds are provided, including stereoisomers, tautomers, and pharmaceutically acceptable salts thereof, useful for inhibiting Btk kinase, and for treating immune disorders such as inflammation mediated by Btk kinase. Methods of using heteroaryl pyridone and aza-pyridone compounds for in vitro, in situ, and in vivo diagnosis, and treatment of such disorders in mammalian cells, or associated pathological conditions, are disclosed.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.