Patent · US Active

Covalent inhibitors of kras G12C

US10273207B2 · kind B2 · utility

24Cited by
53References
34Claims
0Family size

Assignee

Inventors

Key dates

Filing dateFeb 7, 2018
Grant dateApr 30, 2019
Priority date
Expiry dateFeb 7, 2038

Classification

  • Technology area (CPC G)Physics
  • CPC primaryG01N33/58
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Irreversible inhibitors of G12C mutant K-Ras protein are provided. Also disclosed are methods to modulate the activity of G12C mutant K-Ras protein and methods of treatment of disorders mediated by G12C mutant K-Ras protein.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.