Patent · US Active

Phosphatidylinositol 3-kinase inhibitors

US10308639B2 · kind B2 · utility

1Cited by
29References
20Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 10, 2015
Grant dateJun 4, 2019
Priority date
Expiry dateJun 10, 2035

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D513/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present application provides the compounds of formula (J), or pharmaceutically acceptable salts, isomers, tautomer, or a mixture thereof, wherein X, Y, Z, n, m′, A′, R1, R2, and R3 are described herein. The compounds are inhibitors to the activities of phosphatidylinositol 3-kinase (PI3K) and are useful for treating conditions mediated by one or more PI3K isoforms. The present application further provides pharmaceutical compositions that include a compound of formula (I), or pharmaceutically acceptable salts, isomers, tautomer, or mixture thereof, and methods of using these compounds and compositions for treating conditions mediated by one or more PI3K isoforms.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.