Patent · US Active

Bicyclic aryl monobactam compounds and methods of use thereof for the treatment of bacterial infections

US10407421B2 · kind B2 · utility

1Cited by
2References
26Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 2, 2017
Grant dateSep 10, 2019
Priority date
Expiry dateMar 2, 2037

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K31/439
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to bicyclic aryl monobactam compounds of Formula (I), and pharmaceutically acceptable salts thereof, wherein A1, L, M, W, X, Y, Z, RX and Rz are as defined herein. The present invention also relates to compositions which comprise a bicyclic aryl monobactam compound of the invention or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable carrier. The invention further relates to methods for treating a bacterial infection comprising administering to the patient a therapeutically effective amount of a compound of the invention, either alone or in combination with a therapeutically effective amount of one or more beta-lactamase inhibitor compounds.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.