Patent · US Active

Spiropiperidine allosteric modulators of nicotinic acetylcholine receptors

US11332463B2 · kind B2 · utility

1Cited by
6References
54Claims
0Family size

Assignee

Inventors

Key dates

Filing dateApr 29, 2019
Grant dateMay 17, 2022
Priority date
Expiry dateMay 24, 2039

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D513/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present disclosure relates to compounds of formula I that are useful as modulators of 7 nAChR, compositions comprising such compounds, and the use of such compounds for preventing, treating, or ameliorating disease, particularly disorders of the central nervous system such as cognitive impairments in Alzheimer's disease, Parkinson's disease, and schizophrenia, as well as for L-DOPA induced-dyskinesia and inflammation (I).

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.