Patent · US Active

Deuterated pyridone amides and prodrugs thereof as modulators of sodium channels

US11358977B2 · kind B2 · utility

5Cited by
30References
20Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 16, 2018
Grant dateJun 14, 2022
Priority date
Expiry dateJun 16, 2038

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07B2200/05
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Compounds, and pharmaceutically acceptable salts thereof, useful as inhibitors of sodium channels are provided. The compounds have the formula (I) wherein R is H or CH2OPO(OH)2. Also provided are pharmaceutical compositions comprising the compounds or pharmaceutically acceptable salts and methods of using the compounds, pharmaceutically acceptable salts, and pharmaceutical compositions in the treatment of various disorders, including pain.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.