Patent assignee · US · COMPANY

Vertex Pharmaceuticals Incorporated

1,150Patents
816Active
1,150Granted
62Portfolio score

Filing activity: Jul 2, 1990 → Sep 4, 2024 · 316 expiring within 5 years

Most-cited patents

PatentTitleAreaCited byStatus
US5807876A Inhibitors of IMPDH enzyme Chemistry; Metallurgy 191 Expired
US6686193B2 High throughput method and system for screening candidate compounds for activity against target ion channels Physics 186 Expired
US7495103B2 Modulators of ATP-binding cassette transporters Physics 154 Active
US5585397A Sulfonamide inhibitors of aspartyl protease Chemistry; Metallurgy 150 Expired
US7553855B2 Compositions of N-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline-3-carboxamide Chemistry; Metallurgy 142 Active
US6825190B2 Protein kinase inhibitors and uses thereof Chemistry; Metallurgy 135 Expired
US7846951B2 Thiazoles and oxazoles useful as modulators of ATP-binding cassette transporters Chemistry; Metallurgy 128 Active
US7645789B2 Indole derivatives as CFTR modulators Physics 127 Active
US6054472A Inhibitors of IMPDH enzyme Chemistry; Metallurgy 127 Expired
US6784195B2 Pyrazole compositions useful as inhibitors of ERK Chemistry; Metallurgy 126 Expired
US7659268B2 Modulators of ATP-binding cassette transporters Chemistry; Metallurgy 122 Active
US7776905B2 Modulators of ATP-binding cassette transporters Physics 119 Active
US7691902B2 Modulators of ATP-binding cassette transporters Chemistry; Metallurgy 115 Active
US7754739B2 Modulators of CFTR Chemistry; Metallurgy 115 Active
US7598412B2 Modulators of ATP-binding cassette transporters Chemistry; Metallurgy 115 Expired
US7671221B2 Modulators of ATP-Binding Cassette transporters Human Necessities 115 Active
US5192773A Immunosuppressive compounds Chemistry; Metallurgy 114 Expired
US7741321B2 Modulators of ATP-binding cassette transporters Chemistry; Metallurgy 114 Active
US7553671B2 Modular test tube rack Emerging Cross-Sectional Technologies 113 Expired
US7407976B2 Thiazoles and oxazoles useful as modulators of ATP-Binding Cassette transporters Chemistry; Metallurgy 113 Expired
US6664247B2 Pyrazole compounds useful as protein kinase inhibitors Chemistry; Metallurgy 109 Expired
US7973169B2 Modulators of ATP-Binding Cassette transporters Physics 107 Active
US8642609B2 Modulators of ATP-binding cassette transporters Chemistry; Metallurgy 107 Active
US7956052B2 Modulators of ATP-binding cassette transporters Chemistry; Metallurgy 106 Active
US8163772B2 Solid forms of N-[2,4-bis(1,1-dimethylethyl)-5-hydroxypheny1]-1,4-dihydro-4-oxoquinoline-3-carboxamide Chemistry; Metallurgy 106 Active

Source: USPTO / EPO open patent data. Counts and citation impact are objective bibliographic measures.