Patent · US Active

Substituted pyrrolo[1,2-b]pyridazines as bifunctional degraders of interleukin-1 receptor-associated kinases

US11976071B2 · kind B2 · utility

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9References
14Claims
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Key dates

Filing dateAug 18, 2022
Grant dateMay 7, 2024
Priority date
Expiry dateAug 18, 2042

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02A50/30
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present disclosure provides bifunctional compounds of Formula (I), and pharmaceutically acceptable salts, isotopic forms, isolated stereoisomers, or mixtures of stereoisomers thereof, as IRAK4 degraders via ubiquitin proteasome pathway, and method for treating diseases modulated by IRAK4.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.