Patent · US Active

Isoindolinone derivatives as selective allosteric inhibitors of Egfr mutant cancers

US12209091B2 · kind B2 · utility

1Cited by
0References
30Claims
0Family size

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Key dates

Filing dateNov 25, 2020
Grant dateJan 28, 2025
Priority date
Expiry dateSep 30, 2042

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K47/38
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides compounds which are selective allosteric inhibitors of T790M/L858R, T790M/L858R/C797S, L858R, L858R/C797S containing EGFR mutants, their manufacture, pharmaceutical compositions containing them and their use as therapeutically active substances.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.