Patent · US Expired

Pharmaceutically active 6,9-thiaprostacyclin analogs and derivatives thereof

US4291166A · kind A · utility

3Cited by
2References
15Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 13, 1978
Grant dateSep 22, 1981
Priority date
Expiry dateMar 13, 1998

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D333/78
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Stable biologically active 6,9 .alpha.-thiaprostacyclin derivatives having the formula ##STR1## wherein X represents >S, >SO or >SO.sub.2 ; PA1 Y represents (E) and PA2 (Z)-->C.dbd.CH--CH.sub.2 CH.sub.2 CH.sub.2 COOR, PA2 (E)-->CH--CH.dbd.CH--CH.sub.2 CH.sub.2 COOR or >CH--CH.sub.2 --CH.sub.2 --CH.sub.2 --CH.sub.2 COOR; and PA1 R represents hydrogen, a pharmaceutically acceptable cation or a pharmaceutically acceptable lower alkyl group.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.