Kyriacos C. Nicolaou
60Patents
13h-index
116Co-inventors
87Inventor score
Filing activity: Mar 13, 1978 → Mar 18, 2019
Most-cited inventions
| Patent | Title | Area | Cited by | Status |
|---|---|---|---|---|
| US5264586A | Analogs of calicheamicin gamma1I, method of making and using the same | Chemistry; Metallurgy | 141 | Expired |
| US5384412A | Saccharide intermediates in the formation of the calicheamicin and esperamicin oligosaccharides | Chemistry; Metallurgy | 81 | Expired |
| US6380394B1 | Epothilone analogs | Emerging Cross-Sectional Technologies | 54 | Expired |
| US6441186B1 | Epothilone analogs | Chemistry; Metallurgy | 44 | Expired |
| US5552534A | Non-Peptide peptidomimetics | Chemistry; Metallurgy | 30 | Expired |
| US4442099A | Leukotriene analogues | Chemistry; Metallurgy | 29 | Expired |
| US6531497B1 | Epothilone derivatives and their synthesis and use | Emerging Cross-Sectional Technologies | 26 | Expired |
| US4759880A | Alkanoarachidonic acids | Chemistry; Metallurgy | 25 | Expired |
| US6660758B1 | Epothilone analogs | Chemistry; Metallurgy | 21 | Expired |
| US4567290A | Leukotriene analogues | Chemistry; Metallurgy | 21 | Expired |
| US7410998B2 | Inhibitors of NADH:ubiquinone oxidoreductase | Chemistry; Metallurgy | 19 | Expired |
| US5413992A | Daunomycin derivative with reduced cytotoxicity toward normal cells | Chemistry; Metallurgy | 17 | Expired |
| US8071795B2 | HIF inhibitors | Human Necessities | 16 | Active |
| US4977286A | Glycolipids | Chemistry; Metallurgy | 12 | Expired |
| US5281710A | Dynemicin analogs: synthesis, methods of preparation and use | Chemistry; Metallurgy | 8 | Expired |
| US5276159A | Dynemicin analogs: syntheses, methods of preparation and use | Chemistry; Metallurgy | 6 | Expired |
| US5965718A | Analogs of sarcodictyin and eleutherobin | Human Necessities | 5 | Expired |
| US7173137B2 | Epothilone analogs | Chemistry; Metallurgy | 3 | Expired |
| US5183942A | Ten-membered ring enediynediols and enediynediones having DNA cleaving properties | Chemistry; Metallurgy | 3 | Expired |
| US5110949A | Method of synthesizing leukotriene B.sub.4 and derivatives thereof | Chemistry; Metallurgy | 3 | Expired |
| US5527805A | Dynemicin analogs: syntheses, methods of preparation and use | Chemistry; Metallurgy | 3 | Expired |
| US7652033B2 | HIF-1 inhibitors | Chemistry; Metallurgy | 3 | Expired |
| US4291166A | Pharmaceutically active 6,9-thiaprostacyclin analogs and derivatives thereof | Chemistry; Metallurgy | 3 | Expired |
| US4981981A | Sesquiterpene epoxides and process for their preparation | Chemistry; Metallurgy | 3 | Expired |
| US9777013B2 | Derivatives of uncialamycin, methods of synthesis and their use as antitumor agents | Human Necessities | 2 | Active |
Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.