Patent · US Expired

Automated system for polynucleotide synthesis and purification

US5047524A · kind A · utility

235Cited by
7References
10Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 21, 1988
Grant dateSep 10, 1991
Priority date
Expiry dateDec 21, 2008

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC40B60/14
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

A method and system for polynucleotide synthesis and purification are provided which employ solid phase synthesis on a nonswellable porous polystyrene support by phosphoramidite or hydrogen phosphonate chemistries. The polystyrene support gives rise to fewer tritylated failure squences caused by chain growth from extraneous support sites. Consequently, currently used rapid purification techniques depending on trityl hydrophobicity give a more highly purified product. The method and system also employ nucleoside intermediates whose exocyclic amines are protected by base-labile groups which permit simultaneous cleavage and deprotection of the completed polynucleotide chain in the presence of the solid phase support. This latter feature allows practical automation of both the synthesis and purification of polynucleotides.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.