Patent · US Expired

Glycerol derivatives

US5057530A · kind A · utility

5Cited by
1References
5Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 19, 1989
Grant dateOct 15, 1991
Priority date
Expiry dateMay 19, 2009

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D295/088
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Glycerol derivatives of the formula ##STR1## wherein one of the residues R.sup.1, R.sup.2 and R.sup.3 is a group U of the formula OY.sup.1 or --X.sup.1 --CO--(A.sup.1).sub.n --Z.sup.1, another residue is a group V of the formula OY.sup.2 or --X.sup.2 --CO--(A.sup.2).sub.p --Z.sup.2, and the remaining residue is a group W of the formula --X.sup.3 T--(C.sub.2-6 -alkylene)-N.sup.+ R A.sup.- in which one of X.sup.1, X.sup.2 and X.sup.3 is oxygen or NQ.sup.1 and the other two are oxygen and the remaining symbols have the significance given below, and their hydrates are described and are prepared by introducing or generating the residues R.sup.1, R.sup.2 and R.sup.3 in corresponding glycerol derivatives. The compounds of formula I are active as inhibitors of blood platelet activating factor or as inhibitors of the growth of tumors.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.