Patent · US Expired

Novel carboxamide pyridine compounds which have useful pharmaceutical utility

US5084466A · kind A · utility

51Cited by
3References
16Claims
0Family size

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Key dates

Filing dateJan 16, 1990
Grant dateJan 28, 1992
Priority date
Expiry dateJan 16, 2010

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02P20/55
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Novel carboxamides and sulfonamides are described having of the formula EQU R.sup.1 --A--(W).sub.a --X--(CH.sub.2).sub.b --(Y).sub.c --B--Z--COOR (I), in which R.sup.1, A, W, X, Y, B, Z, R, a, b and c are as provided in the description. These compounds are useful in the treatment of thromboses, apoplexy, myocardial infarct, inflammations, arteriosclerosis as well as in the treatment and prevention of tumors. These novel compounds are prepared by eliminating the protective groups in corresponding compounds with protected amidino or guanidino groups.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.