Substituted 2-carboxylindoles having pharmaceutical activity
US5145845A · kind A · utility
23Cited by
6References
16Claims
0Family size
Assignee
Inventors
Key dates
| Filing date | May 14, 1991 |
| Grant date | Sep 8, 1992 |
| Priority date | — |
| Expiry date | May 14, 2011 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D403/06
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
The present invention relates to novel compounds, which are derivatives of ureas, thioureas, carbamates, sulfonylureas, sulfonamides, amides, and thioamides of 2-carboxyindoles as illustrated by the formula ##STR1## The invention also relates to methods for the preparation of the novel compounds, as well as to pharmaceutical compositions or methods of use for the novel compounds. More specifically, the compounds of the present invention are useful in the treatment of neurodegenerative disorders including cerebrovascular disorders as well as in the treatment of schizophrenia or epilepsy; and as analgesics and anxiolytics.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.