Inventor · Irvine, CA, US

Thomas C. Malone

80Patents
12h-index
72Co-inventors
87Inventor score

Filing activity: Mar 13, 1989 → Sep 10, 2018

Most-cited inventions

PatentTitleAreaCited byStatus
US6765012B2 3-(Arylamino)methylene-1,3-dihydro-2H-indol-2-ones as kinase inhibitors Chemistry; Metallurgy 84 Expired
US8512738B2 Biodegradable intravitreal tyrosine kinase implants Human Necessities 58 Active
US8409607B2 Sustained release intraocular implants containing tyrosine kinase inhibitors and related methods Emerging Cross-Sectional Technologies 53 Active
US7771742B2 Sustained release intraocular implants containing tyrosine kinase inhibitors and related methods Emerging Cross-Sectional Technologies 37 Active
US6458781B1 Substituted diarylalkyl amides as calcium channel antagonists Chemistry; Metallurgy 37 Expired
US6541504B1 (3Z)-3-(2,3-dihydro-1H-inden-1-ylidene)-1,3-dihydro-2H-indol-2-ones as kinase inhibitors Chemistry; Metallurgy 32 Expired
US6747025B1 Kinase inhibitors for the treatment of disease Chemistry; Metallurgy 30 Expired
US5145845A Substituted 2-carboxylindoles having pharmaceutical activity Chemistry; Metallurgy 23 Expired
US7015220B2 3-(arylamino)methylene-1, 3-dihydro-2H-indol-2-ones as kinase inhibitors Chemistry; Metallurgy 21 Expired
US8968766B2 Sustained release intraocular implants containing tyrosine kinase inhibitors and related methods Emerging Cross-Sectional Technologies 19 Active
US7060844B2 (3Z)-3-(2,3-dihydro-1H-inden-1-ylidene)-1,3-dihydro-2H-indol-2-ones as kinase inhibitors Chemistry; Metallurgy 16 Expired
US6423689B1 Peptidyl calcium channel blockers Human Necessities 15 Expired
US5002950A 7-deazaguanines as immunomodulators Chemistry; Metallurgy 12 Expired
US6117841A Substituted peptidylamine calcium channel blockers Human Necessities 12 Expired
US7125908B2 Treating pain using selective antagonists of persistent sodium current Human Necessities 11 Expired
US4921858A 7-deazaguanines as immunomodulators Chemistry; Metallurgy 10 Expired
US7060723B2 Treating neurological disorders using selective antagonists of persistent sodium current Human Necessities 9 Expired
US6197771A Glutamate (ampa/kainate) receptor antagonists: N-substituted fused azacycloalkylquinoxalinediones Chemistry; Metallurgy 7 Expired
US7767718B2 Treating pain using selective antagonists of persistent sodium current Human Necessities 6 Active
US7915443B2 Sulfoximines as kinase inhibitors Chemistry; Metallurgy 5 Active
US7749530B2 Kinase inhibitors Chemistry; Metallurgy 4 Active
US7705055B2 Treating neurological disorders using selective antagonists of persistent sodium current Human Necessities 4 Active
US9433631B2 4-pregenen-11β-17-21-triol-3,20-dione derivatives Human Necessities 3 Active
US7977351B2 Heteroaryl dihydroindolones as kinase inhibitors Chemistry; Metallurgy 3 Active
US9371314B2 Pyridyl benzothiophenes as kinase inhibitors Chemistry; Metallurgy 3 Active

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.