Patent · US Expired

TGF-B compositions and method

US5147854A · kind A · utility

10Cited by
3References
16Claims
0Family size

Assignee

Inventor

Key dates

Filing dateMay 22, 1990
Grant dateSep 15, 1992
Priority date
Expiry dateMay 22, 2010

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P35/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Transforming growth factor-beta (TGF-beta) is enhanced in its therapeutic activity by utilizing it in combination with a synergistic effective amount of a polyunsaturated fatty acid (PUFA). In a preferred embodiment, type 1 transforming growth factor beta (TGF-.sym.1) exhibits enhanced anti-neoplastic activity when utilized in combination with an n=3 or n=6 polyunsaturated fatty acid. Examples of suitable unsaturated fatty acids include linoleic, alpha-linolenic, arachidonic, gamma-linolenic, dihomogammalinolenic, eicosapentaenoic and docosahexaenoic. Combinations of these agents effectively kill various human carcinoma and melanoma cell lines under defined conditions in vitro at picomolar concentrations of TGF-.beta.1 and at .mu.g/ml concentrations of the polyunsaturated fatty acid, levels where the respective two agents acting alone are ineffective.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.