Patent · US Expired

Camptothecin analogs as potent inhibitors of topoisomerase I

US5244903A · kind A · utility

56Cited by
6References
1Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 22, 1990
Grant dateSep 14, 1993
Priority date
Expiry dateOct 22, 2010

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D491/22
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A method for synthesizing camptothecin analogs using a novel hydroxyl-containing tricyclic intermediate and the camptothecin analogs produced by the process. The camptothecin analogs are effective inhibitors of topoisomerase.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.