Benzodiazepine derivatives, compositions containing them and their use in therapy
US5410049A · kind A · utility
13Cited by
2References
6Claims
0Family size
Assignee
Inventor
Key dates
| Filing date | Dec 17, 1992 |
| Grant date | Apr 25, 1995 |
| Priority date | — |
| Expiry date | Dec 17, 2012 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D409/12
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
Compounds of formula (I), and salts and prodrugs thereof ##STR1## wherein: R.sup.1 is H, certain optionally substituted C.sub.1-6 alkyl, or C.sub.3-7 cyclocalkyl; PA1 R.sup.2 represents a group ##STR2## wherein X is O, S or NR.sup.8 where R.sup.8 is H or C.sub.1-4 alkyl; R.sup.3 is C.sub.1-6 alkyl, halo or NR.sup.6 R.sup.7 ; PA1 R.sup.4 is C.sub.1-7 alkyl, C.sub.3-7 cycloalkyl, C.sub.4-7 cycloalkylalkyl or optionally substituted aryl; PA1 n is 0, 1, 2 or 3; are CCK and/or gastrin receptor antagonists. They and compositions thereof are useful in therapy.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.