Patent · US Expired

Substituted aryl piperazines as neurokinin antagonists

US5607936A · kind A · utility

24Cited by
6References
12Claims
0Family size

Assignee

Inventors

Key dates

Filing dateSep 30, 1994
Grant dateMar 4, 1997
Priority date
Expiry dateSep 30, 2014

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D495/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Disclosed are substituted aryl piperazines of Formula I ##STR1## are tachykinin receptor antagonists useful in the treatment of inflammatory diseases, pain or migraine, asthma and emesis. In particular compounds of Formula I are shown to be neurokinin antagonists.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.