Inventor · Freehold, NJ, US

Malcolm MacCoss

117Patents

28h-index

239Co-inventors

93Inventor score

Filing activity: Feb 3, 1982 → Sep 24, 2021

Most-cited inventions

Patent	Title	Area	Cited by	Status
US7125855B2	Nucleoside derivatives as inhibitors of RNA-dependent RNA viral polymerase	Emerging Cross-Sectional Technologies	214	Expired
US6777395B2	Nucleoside derivatives as inhibitors of RNA-dependent RNA viral polymerase of hepatitis C virus	Emerging Cross-Sectional Technologies	212	Expired
US7105499B2	Nucleoside derivatives as inhibitors of RNA-dependent RNA viral polymerase	Emerging Cross-Sectional Technologies	155	Expired
US6699871B2	Beta-amino heterocyclic dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes	Chemistry; Metallurgy	140	Expired
US7879815B2	Nucleoside aryl phosphoramidates for the treatment of RNA-dependent RNA viral infection	Human Necessities	100	Active
US5719147A	Morpholine and thiomorpholine tachykinin receptor antagonists	Chemistry; Metallurgy	83	Expired
US5691336A	Morpholine compounds are prodrugs useful as tachykinin receptor antagonists	Chemistry; Metallurgy	79	Expired
US4579849A	N-alkylguanine acyclonucleosides as antiviral agents	Chemistry; Metallurgy	71	Expired
US6372733B1	Hexahydro-5-imino-1,4-1,4-thiazepine derivatives as inhibitors of nitric oxide synthases	Chemistry; Metallurgy	62	Expired
US6166037A	Pyrrolidine and piperidine modulators of chemokine receptor activity	Chemistry; Metallurgy	57	Expired
US7534767B2	C-purine nucleoside analogs as inhibitors of RNA-dependent RNA viral polymerase	Chemistry; Metallurgy	50	Expired
US7632821B2	Ribonucleoside cyclic acetal derivatives for the treatment of RNA-dependent RNA viral infection	Chemistry; Metallurgy	48	Active
US5430128A	Peptidyl derivatives as inhibitors of interleukin-1.beta. converting enzyme	Human Necessities	45	Expired
US5434248A	Peptidyl derivatives as inhibitors of interleukin-1.beta. converting enzyme	Chemistry; Metallurgy	45	Expired
US5750549A	Cycloalkyl tachykinin receptor antagonists	Chemistry; Metallurgy	44	Expired
US5629322A	Cyclic amidine analogs as inhibitors of nitric oxide synthase	Chemistry; Metallurgy	42	Expired
US5057517A	Piperazinyl derivatives of purines and isosteres thereof as hypoglycemic agents	Chemistry; Metallurgy	39	Expired
US5962462A	Spiro-substituted azacycles as modulators of chemokine receptor activity	Chemistry; Metallurgy	37	Expired
US4471113A	Prodrugs based on phospholipid-nucleoside conjugates	Chemistry; Metallurgy	36	Expired
US5877191A	Phenyl spiroethercycloalkyl tachykinin receptor antagonists	Chemistry; Metallurgy	35	Expired
US5229381A	Substituted azetidinones as anti-inflammatory and antidegenerative agents	Chemistry; Metallurgy	34	Expired
US6136827A	Cyclic amine modulations of chemokine receptor activity	Chemistry; Metallurgy	33	Expired
US5348953A	Substituted azetidinones as anti-inflammatory and antidegenerative agents	Chemistry; Metallurgy	32	Expired
US5292726A	N,N-diacylpiperazines	Chemistry; Metallurgy	31	Expired
US5512570A	Treatment of emesis with morpholine tachykinin receptor antagonists	Chemistry; Metallurgy	31	Expired

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.