Patent · US Expired

Prodrugs for enzyme mediated activation

US5621002A · kind A · utility

103Cited by

0References

9Claims

0Family size

Assignees

Behringwerke Aktiengesellschaft · DE
Laboratories Hoechst S/A · FR

Inventors

Klaus Bosslet · Marburg, DE
J org Czech · Marburg, DE
Dieter Hoffmann · Marburg, DE
Andrea Vasella · Zürich, CH
Roland Hoos · Sierre, CH
François Tillequin · Paris, FR
Jean-Claude Florent · Boulogne-Billancourt, FR
Michel Azoulay · Richibucto, CA
Claude Monneret · Paris, FR
Jean-Claude Jacquesy · Guéret, FR
Jean-Pierre Gesson · Poitiers, FR
Michel Koch · La Celle-Saint-Cloud, FR

Key dates

Filing date	Sep 9, 1994
Grant date	Apr 15, 1997
Priority date	—
Expiry date	Sep 9, 2014

Classification

Technology area (CPC B)Performing Operations; Transporting
CPC primaryB82Y5/00
WIPO fieldPharmaceuticals
WIPO sectorChemistry

Abstract

Enzymatically clearable prodrugs with reduced Michaelis-Menten constant (Km) are described.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.